| Bioactivity | Sheng Gelieting (CGT-8012) is a dipeptidy peptidase-IV enzyme (DP-IV) inhibitor. Sheng Gelieting has great DP-IV inhibition activity with an IC50 value of 87 nM. Sheng Gelieting can be used for curing or preventing diseases relevant to the dipeptidy peptidase-IV enzyme, such as the diabetes, particularly the II-type diabete[1]. |
| Target | IC50: 87 nM (DP-IV) |
| Invitro | Sheng Gelieting has great dipeptidy peptidase-IV enzyme (DP-IV) inhibition activity with an IC50 value of 87 nM[1]. |
| Name | Sheng Gelieting |
| CAS | 1152810-23-5 |
| Formula | C17H16F6N4O |
| Molar Mass | 406.33 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Qiang Yu, et al. Beta-amino tetrahydropyrazine, tetrahydropyrimidine and tetrahydropyridine used as dipeptidy peptidase inhibitors for curing or preventing diabetes. Patent. CN101899047A. |