| Bioactivity | Setin-1 is one of the most potent inhibitors of Set7, acting by inhibiting KMTase G9a[1]. |
| CAS | 1313802-67-3 |
| Formula | C29H21F3N2O2 |
| Molar Mass | 486.48 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Kashyap S, et al. Using 'biased-privileged' scaffolds to identify lysine methyltransferase inhibitors. Bioorg Med Chem. 2014 Apr 1;22(7):2253-60. |