| Bioactivity | Setastine (EGIS-2062 (free acid); EGYT-2062 (free acid) is an orally effective, non-sedative and long acting anti-allergic agent. Setastine possesses potent histamine Hi-receptor blocking properties and can be used for allergies and rhinitis research[1]<. |
| Target | IC50:Histamine Hi-receptor |
| Name | Setastine |
| CAS | 64294-95-7 |
| Formula | C22H28ClNO |
| Molar Mass | 357.92 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Németh, A., & Huszti, Z. (1988). The effect of a new antihistamine drug, Loderix® (EGIS-2062), on stimulus-evoked histamine release from rat peritoneal mast cells. Agents and Actions, 23(3-4), 194–197. |