| Bioactivity | ST-2560 is a selective inhibitor of the NaV1.7 sodium channel with IC50 at 39 nM. ST-2560 can be used to study pain behavior and cardiovascular models[1]. |
| In Vivo | ST-2560 (0.1-0.3 mg/kg, 皮下注射) 在非人灵长类动物 (NHP) 行为模型中可抑制有害的机械和化学诱发反射[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
| Formula | C27H34N10O4 |
| Molar Mass | 562.62 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Mulcahy JV, et al. ST-2560, a selective inhibitor of the NaV1.7 sodium channel, affects nocifensive and cardiovascular reflexes in non-human primates. Br J Pharmacol. 2024 May 7. |