Bioactivity | SOS1-IN-16 (Comp 54) is a selective inhibitor of SOS1 with an IC50 of 7.2 nM. SOS1-IN-16 has inhibitory activity of CYP3A4 when using testosterone as a substrate, with an IC50 of 8.9μM. SOS1-IN-16 can be used for cancer research[1]. |
Name | SOS1-IN-16 |
CAS | 2930763-85-0 |
Formula | C30H31F3N4O3 |
Molar Mass | 552.59 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Chen SJ, et.al.Polysubstituted benzazepine heteroaryl derivative and application thereof |