Bioactivity | SN05 is a potent amino acid transport (AAT) inhibitor with Kis of 2.77 μM, 0.73 μM, 0.87 μM, 3.7 μM, 7.25 μM, 7.23 μM and 2.22 μM for human ASCT1, rat ASCT2, human ASCT2, EAAT1, EAAT2, EAAC1 and EAAT5, respectively. SN05 can be used for researching anticancer[1]. |
Target | Ki: 2.77 μM (human ASCT1), 0.73 μM (rat ASCT2), 0.87 μM (human ASCT2), 3.7 μM (EAAT1), 7.25 μM (EAAT2), 7.23 μM (EAAC1), 2.22 μM (EAAT5) |
Name | SN05 |
CAS | 2768663-51-8 |
Formula | C18H17NO4 |
Molar Mass | 311.33 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Christof GREWER, et al. Inhibitors of amino acid transport. WO2022087630A1 |