| Bioactivity | SIK2-IN-1 (compound 8g) is a potent SIK2 inhibitor over other AMPK kinases. SIK2-IN-1 exhibits favorable in vitro ADMET profiles and decent cellular activities[1]. |
| Target | SIK2 |
| Name | SIK2-IN-1 |
| Formula | C25H28F3N7O2S |
| Molar Mass | 547.60 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Zhu W, et al. Discovery of novel and selective SIK2 inhibitors by the application of AlphaFold structures and generative models. Bioorg Med Chem. 2023 Jul 13;91:117414. |