| Bioactivity | SHU 9119 is a potent human melanocortin 3 and 4 receptors (MC3/4R) antagonist and a partial MC5R agonist; with IC50 values of 0.23, 0.06, and 0.09 nM for human MC3R, MC4R and MC5R, respectively. | ||||||
| Name | SHU 9119 | ||||||
| CAS | 168482-23-3 | ||||||
| Sequence | Ac-{Nle}-cyclo[Asp-His-D-{Nal}-Arg-Trp-Lys]-NH2 | ||||||
| Shortening | Ac-{Nle}-cyclo[DHD-{Nal}-RWK]-NH2 | ||||||
| Formula | C54H71N15O9 | ||||||
| Molar Mass | 1074.24 | ||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||
| Storage | Sealed storage, away from moisture and light
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light) |