| Bioactivity | SGC2085 hydrochloride is a potent and selective inhibitor of coactivator associated arginine methyltransferase 1 (CARM1) with an IC50 of 50 nM. SGC2085 hydrochloride also selectively inhibits PRMT6 with an IC50 value of 5.2 μM, but not other PRMT proteins[1]. |
| Invitro | SGC2085 hydrochloride (1 μM, 10 μM, 50 μM；48 h) 对 21 种人类蛋白质甲基转移酶的具有完全选择性[1]。SGC2085 hydrochloride (10 μM；48 h) 表现出低细胞渗透性，在 HEK293 细胞中无细胞活性[1]。 |
| Name | SGC2085 hydrochloride |
| CAS | 1821908-49-9 |
| Formula | C19H25ClN2O2 |
| Molar Mass | 348.87 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
SGC2085 hydrochloride
CAS: 1821908-49-9 F: C19H25ClN2O2 W: 348.87
SGC2085 hydrochloride is a potent and selective inhibitor of coactivator associated arginine methyltransferase 1 (CARM1)
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