| Bioactivity | SGC-STK17B-1 is an ATP-competitive and selective STK17B inhibitor (IC50: 34 nM, KD: 5.6 nM)[1]. |
| Target | 34 nM (STK17B). |
| Name | SGC-STK17B-1 |
| CAS | 2650530-00-8 |
| Formula | C16H10N2O2S3 |
| Molar Mass | 358.46 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Picado A, et al. A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation. J Med Chem. 2020 Dec 10;63(23):14626-14646. |