Bioactivity | SER-601 is a potent and selective peripheral cannabinoid (CB2) receptor agonist with a Ki of 6.3 nM. SER-601 has analgesic and antidiabetic properties and can be used for relevant research[1]. |
In Vivo | SER-601 (1, 3 mg/kg, i.p.) 在小鼠福尔马林实验中展现出剂量依赖性的镇痛作用[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. |
CAS | 1048038-90-9 |
Formula | C28H38N2O2 |
Molar Mass | 434.61 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Pasquini S, et al. Investigations on the 4-quinolone-3-carboxylic acid motif. 2. Synthesis and structure-activity relationship of potent and selective cannabinoid-2 receptor agonists endowed with analgesic activity in vivo. J Med Chem. 2008 Aug 28;51(16):5075-84. |