| Bioactivity | PD-135666 is a dipeptide that inhibits the cholecystokinin B (CCK B) receptor more than the CCK A receptor. PD-135666 binds to CCK B receptors with an IC50 of 0.1 nM in mouse cerebral cortex, whereas its enantiomer PD-140548 preferentially binds to CCK A receptors with an IC50 of 2.8 nM in rat pancreas. PD-135666 exhibits anxiolytic effects in animal models[1]. |
| Target | CCK B receptor |
| CAS | 138828-39-4 |
| Formula | C30H35NO6S |
| Molar Mass | 537.67 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |