Bioactivity | Rivulariapeptolides 988 is a high potent and selective serine protease inhibitor with IC50 values of 95.46 nM, 15.29 nM and 85.50 nM for chymotrypsin, elastase and proteinase K, respectively[1]. |
Target | IC50: 95.46 nM (chymotrypsin); 15.29 nM (elastase) and 85.50 nM (proteinase K). |
Invitro | Rivulariapeptolides 998 (0-3 μM, 40 min) has high potency and distinct selectivity with IC50 values of 95.46 nM, 15.29 nM and 85.50 nM for chymotrypsin, elastase and proteinase K, respectively[1]. |
Name | Rivulariapeptolides 988 |
Formula | C50H68N8O13 |
Molar Mass | 989.12 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Raphael Reher, et al. Native metabolomics identifies the rivulariapeptolide family of protease inhibitors. Nat Commun. 2022 Aug 8;13(1):4619. |