Rivulariapeptolides 1185

CAS: F: C61H87N9O15 W: 1186.39

Rivulariapeptolides 1185 is a high potent and selective serine protease inhibitor with IC50 values of 13.17 nM, 23.59 nM

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Bioactivity	Rivulariapeptolides 1185 is a high potent and selective serine protease inhibitor with IC50 values of 13.17 nM, 23.59 nM and 55.26 nM for chymotrypsin, elastase and proteinase K, respectively[1].
Target	IC50: 13.17 nM (chymotrypsin); 23.59 nM (elastase) and 55.26 nM (proteinase K).
Invitro	Rivulariapeptolides 1185 (0-3 μM, 40 min) has high potency and distinct selectivity with IC50 values of 13.17 nM, 23.59 nM and 55.26 nM for chymotrypsin, elastase and proteinase K, respectively[1].
Name	Rivulariapeptolides 1185
Formula	C61H87N9O15
Molar Mass	1186.39
Transport	Room temperature in continental US; may vary elsewhere.
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.
Reference	[1]. Raphael Reher, et al. Native metabolomics identifies the rivulariapeptolide family of protease inhibitors. Nat Commun. 2022 Aug 8;13(1):4619.