Bioactivity | Rivulariapeptolides 1121 is a high potent and selective serine protease inhibitor with IC50 values of 35.52 nM, 13.24 nM and 48.05 nM for chymotrypsin, elastase and proteinase K, respectively[1]. |
Target | IC50: 35.52 nM (chymotrypsin); 13.24 nM (elastase) and 48.05 nM (proteinase K). |
Invitro | Rivulariapeptolides 1121 (0-3 μM, 40 min) has high potency and distinct selectivity with IC50 values of 35.52 nM, 13.24 nM and 48.05 nM for chymotrypsin, elastase and proteinase K, respectively[1]. |
Name | Rivulariapeptolides 1121 |
Formula | C56H83N9O15 |
Molar Mass | 1122.31 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Raphael Reher, et al. Native metabolomics identifies the rivulariapeptolide family of protease inhibitors. Nat Commun. 2022 Aug 8;13(1):4619. |