| Bioactivity | RY796 is a potent and selective voltage-gated potassium (KV2) channel inhibitor with IC50s of 0.25 μM and 0.09 μM for KV2.1 and KV2.2. RY796 has analgesic activity[1]. | ||||||||||||
| Target | IC50: 0.25 μM (KV2.1) and 0.09 μM (KV2.2) | ||||||||||||
| Name | RY796 | ||||||||||||
| CAS | 1393441-53-6 | ||||||||||||
| Formula | C21H27N3O2 | ||||||||||||
| Molar Mass | 353.46 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Herrington J, et al. Identification of novel and selective Kv2 channel inhibitors. Mol Pharmacol. 2011 Dec;80(6):959-64. |