Bioactivity | RXFP1 receptor agonist-1 (Example 2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-1 inhibits cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 300 nM[1]. |
Name | RXFP1 receptor agonist-1 |
CAS | 2924619-64-5 |
Formula | C31H29F7N2O4 |
Molar Mass | 626.56 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Donald J.P. Pinto, et al. Rxfp1 modulators for the treatment of heart failure. Patent. WO2023077041A1. |