Bioactivity | RIPK-IN-4 is a potent and selective RIPK2 inhibitor with excellent oral bioavailability, and has an IC50 of 3 nM[1]. | ||||||||||||
Target | IC50: 3 nM (RIPK2) | ||||||||||||
Name | RIPK-IN-4 | ||||||||||||
CAS | 2141969-56-2 | ||||||||||||
Formula | C18H21FN4O3S | ||||||||||||
Molar Mass | 392.45 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. He X, et al. Identification of Potent and Selective RIPK2 Inhibitors for the Treatment of Inflammatory Diseases. ACS Med Chem Lett. 2017 Sep 27;8(10):1048-1053. |