Bioactivity | RGB097 is a potent D-dopachrome tautomerase (D-DT) inhibitor with an IC50 value of 0.5 µM. RGB097 has the potential for the research of cancer[1]. |
Target | IC50: 0.5 µM (D-DT) |
Formula | C26H22F3N5O3 |
Molar Mass | 509.48 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Angelina Osipyan, et al. The synthesis of 1,2,3-triazoles as binders of D-dopachrome tautomerase (D-DT) for the development of dual-targeting inhibitors. European Journal of Medicinal Chemistry. 2024, 276: 116665. |