| Bioactivity | RBP4 inhibitor 1 (compound 43b) is a potent and orally active retinol-binding protein 4 (RBP4) inhibitor with IC50s of 28 nM and 110 nM for human and mouse RBP4. RBP4 inhibitor 1 has a potent and long-lasting blood RBP4-level-reducing effect in mice[1]. |
| Target | IC50: 28 nM (human RBP4) and 110 nM (mouse RBP4) |
| Name | RBP4 inhibitor 1 |
| CAS | 1198180-03-8 |
| Formula | C14H13F6NO3 |
| Molar Mass | 357.25 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Shinji Nakamura, et al. Discovery of phenylpyrrolidine derivatives as a novel class of retinol binding protein 4 (RBP4) reducers. Bioorg Med Chem. 2022 Jan 15;54:116553. |
RBP4 inhibitor 1
CAS: 1198180-03-8 F: C14H13F6NO3 W: 357.25
RBP4 inhibitor 1 (compound 43b) is a potent and orally active retinol-binding protein 4 (RBP4) inhibitor with IC50s of 2
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