Bioactivity | RARα antagonist 1 (compound 21) is an orally active and selective retinoic acid receptor α(RARα) antagonist, with the IC50 of 4.6nM[1]. |
Target | 4.6nM (RARα) |
Name | RARα antagonist 1 |
Formula | C26H23NO4 |
Molar Mass | 413.47 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Al Noman MA, et al. Strategies for developing retinoic acid receptor alpha-selective antagonists as novel agents for male contraception [published online ahead of print, 2023 Sep 25]. Eur J Med Chem. 2023;261:115821. |