| Bioactivity | R-84760 is a selective κ-opioid receptor agonist. R-84760 has antinociceptive effect[1][2]. |
| Invitro | 在豚鼠脑膜部分的阿片受体结合试验中，R-84760 对 κ-阿片受体的亲和力比 CI-977 (HY-105235) 高 5 倍，R-84760 对 κ-阿片受体的选择性高于 U-69593 (HY-12363)[1]。 MCE has not independently confirmed the accuracy of these methods. They are for reference only. 0 --> R-84760 相关抗体: |
| CAS | 157824-23-2 |
| Formula | C19H25Cl3N2OS |
| Molar Mass | 435.84 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Fujibayashi K, et al. Pharmacological properties of R-84760, a novel kappa-opioid receptor agonist.[J].European Journal of Pharmacology, 1994, 261(1-2):133-140. [2]. Fujibayashi K, et al. Profiles of the antinociceptive effect of R-84760, a selective kappa-opioid receptor agonist, in the formalin test in mice. Jpn J Pharmacol. 1995 May;68(1):57-63. |