| Bioactivity | Quercetagetin (6-Hydroxyquercetin) is a flavonoid[1]. Quercetagetin is a moderately potent and selective, cell-permeable pim-1 kinase inhibitor (IC50, 0.34 μM)[2]. Anti-inflammatory and anticancer properties. | ||||||||||||
| Invitro | Quercetagetin also inhibits PIM2, PKA, and RSK2 with IC50s of 3.45, 21.2, and 2.82 µM, respectively[2].Quercetagetin (0.1, 1, 10, and 100 μM, 72 hours) inhibits growth of RWPE2 prostate cancer cells with average ED50 is 3.8 μM[2]. Cell Viability Assay[2] Cell Line: | ||||||||||||
| Name | Quercetagetin | ||||||||||||
| CAS | 90-18-6 | ||||||||||||
| Formula | C15H10O8 | ||||||||||||
| Molar Mass | 318.24 | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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