| Bioactivity | Protease-Activated Receptor-4 is the agonist of proteinase-activated receptor-4 (PAR4). | ||||||
| Invitro | GYPGKF-NH2 significantly reduces the agonistic potency of AYPGKF-NH2 by 25-fold[1]. GYPGKF-NH2 (500 μM) does not cause contraction or relaxation of the guinea pig IAS strips[2]. | ||||||
| Name | Protease-Activated Receptor-4 | ||||||
| CAS | 245443-52-1 | ||||||
| Sequence | Gly-Tyr-Pro-Gly-Lys-Phe-NH2 | ||||||
| Shortening | GYPGKF-NH2 | ||||||
| Formula | C33H46N8O7 | ||||||
| Molar Mass | 666.77 | ||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||
| Storage | Sealed storage, away from moisture
*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) |