| Bioactivity | Plm IV inhibitor-1 (compound 6) is a potent plasmepsin IV (Plm IV) inhibitor with IC50s of 4.1, 0.80, 0.25, 0.35 µM for Plm I, Plm II, Plm IV, Cat D, respectively[1]. |
| Target | IC50: 4.1 µM (Plm I); 0.80 µM (Plm II); 0.25 µM (Plm IV); 0.35 µM (Cat D) |
| Name | Plm IV inhibitor-1 |
| CAS | 1539276-41-9 |
| Formula | C37H51N5O3 |
| Molar Mass | 613.83 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Jaudzems K, et al. Plasmepsin inhibitory activity and structure-guided optimization of a potent hydroxyethylamine-based antimalarial hit. ACS Med Chem Lett. 2014 Jan 13;5(4):373-7. |
Plm IV inhibitor-1
CAS: 1539276-41-9 F: C37H51N5O3 W: 613.83
Plm IV inhibitor-1 (compound 6) is a potent plasmepsin IV (Plm IV) inhibitor with IC50s of 4.1, 0.80, 0.25, 0.35 µM for
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This product is for research use only, not for human use. We do not sell to patients.