| Bioactivity | Pitofenone hydrochloride, a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes and from electric eel with Kis of 36 and 45 μM, respectively. |
| Target | Ki: 36 μM (AChE, bovine erythrocytes), 45 μM (AChE, electric eel) |
| Name | Pitofenone hydrochloride |
| CAS | 1248-42-6 |
| Formula | C22H26ClNO4 |
| Molar Mass | 403.90 |
| Appearance | Solid |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | 4°C, sealed storage, away from moisture *In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture) |
| Reference | [1]. Punekar NS, et al. Acetylcholinesterase inhibition by pitofenone: a spasmolytic compound. Biotechnol Appl Biochem. 1991 Dec;14(3):378-82. |