| Bioactivity | Pipamperone (Floropipamide; McN-JR 3345) dihydrochloride is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and D4 receptor (pKi=8.0) and a low-affinity antagonist of D2 receptor (pKi=6.7)[1]. |
| Target | PAR2, PAR4 |
| Name | Pipamperone dihydrochloride |
| CAS | 2448-68-2 |
| Formula | C21H32Cl2FN3O2 |
| Molar Mass | 448.40 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Erik Buntinx, MD, et al. Selective Serotonergic Properties of Low-Dose Pipamperone May Enhance Antidepressant Effect: Preclinical Evidence. |
Pipamperone dihydrochloride
CAS: 2448-68-2 F: C21H32Cl2FN3O2 W: 448.40
Pipamperone (Floropipamide; McN-JR 3345) dihydrochloride is a high-affinity antagonist of 5-HT2A receptor (pKi=8.2) and
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