Bioactivity | Picrotoxinin (Standard) is the analytical standard of Picrotoxinin. This product is intended for research and analytical applications. Picrotoxinin, a potent convulsant, is a chloride channel blocker. Picrotoxinin is a noncompetitive GABAA receptor antagonist, which negatively modulates the action of GABA on GABAA receptors. Picrotoxinin inhibits α1β2γ2L GABAA receptor with an IC50 of 1.15 μM. |
CAS | 17617-45-7 |
Formula | C15H16O6 |
Molar Mass | 292.28 |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |