| Bioactivity | Phelorphan is a purine MTH1 inhibitor identified through chemical array screening. Although it targets cellular MTH1, its cytotoxicity to cancer cells is weaker than that of other reported inhibitors. The cytotoxicity of MTH1 inhibitors may be attributed to off-target effects, and MTH1 is not essential for cancer cell survival. |
| CAS | 110871-16-4 |
| Formula | C20H22N2O4S |
| Molar Mass | 386.46 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Synthesis of enkephalinase B inhibitors, and their activity on isolated enkephalin-degrading enzymes |
Phelorphan
CAS: 110871-16-4 F: C20H22N2O4S W: 386.46
Phelorphan is a purine MTH1 inhibitor identified through chemical array screening. Although it targets cellular MTH1, it
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