| Bioactivity | Pancreatic lipase/Carboxylesterase 1-IN-1 (Compound 39) is a potent dual inhibitor of pancreatic lipase (PL) and human carboxylesterase 1A (hCES1A) with IC50 values of 2.13 µM and 0.055 µM against PL and hCES1A[1]. |
| Target | IC50: 0.055 µM (hCES1A), 2.13 µM (PL), 6.02 µM (hCES2A) |
| Name | Pancreatic lipase/Carboxylesterase 1-IN-1 |
| CAS | 194235-21-7 |
| Formula | C30H44O4 |
| Molar Mass | 468.67 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Zhang J, et al. Discovery of triterpenoids as potent dual inhibitors of pancreatic lipase and human carboxylesterase 1. J Enzyme Inhib Med Chem. 2022 Dec;37(1):629-640. |