Bioactivity | PROTAC GSPT1 degrader-2 (compound A) is a GSPT1 molecule glue with more than 95% degradation. GSPT1 degrader-8 inhibits cell viability in HL-60 cells with an IC50 of 10 nM[1]. |
CAS | 3024909-61-0 |
Formula | C38H38ClN7O5 |
Molar Mass | 708.21 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Lichao FANG, et al. Gspt1 degraders, compositions comprising the degrader, and methods of using the same. French, WO2024073871A1. 2024-04-11 |