Bioactivity | PROTAC ERα Degrader-8 (compound ii-56) is a potent PROTAC degrader of Erα, with DC50 of 0.000006 μM in MCF7 cells[1]. |
CAS | 3025533-68-7 |
Formula | C47H51N5O4 |
Molar Mass | 749.94 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Relay Therapeutics, Inc. Preparation of bifunctional compounds as estrogen receptor alpha degraders and use thereof. World Intellectual Property Organization, WO2024006781 A1 2024-01-04 |