Bioactivity | PROTAC DYRK2 degrader 1 (compound CP134) is a PROTAC degrader of DYRK2 (Red: DYRK2 inhibitor(HY-161598), black: linker (HY-42776), Blue: E3 ligase ligand (HY-10984))[1]. |
Formula | C42H43Br2N5O9 |
Molar Mass | 921.63 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Jian Chen, et al.Discovery of the First Potent DYRK2 Proteolysis Targeting Chimera Degraders. ACS Med. Chem. Lett. 2024, 15, 5, 659–666. |