Bioactivity | PROTAC BRM/BRG1 degrader-2 (Example.004) is a PROTAC BRM/BRG1 degrader (DC50: < 10 nM in A549 cell; IC50: 15 nM for A549). Blue: E3 ligase ligand (HY-112078), Black: linker (HY-168249), Pink: BRM/BRG1 inhibitor (HY-168248)[1]. |
CAS | 2933124-32-2 |
Formula | C50H60N12O5S |
Molar Mass | 941.15 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Gu Peng. Brm selective degradation agent compound and use thereof. Patent. WO2023093728 |