| Bioactivity | PROTAC BRM/BRG1 degrader-1 (Example 253) is a PROTAC BRM/BRG1 degrader, with DC50 of 10-100 nM for BRM, > 1 μM for BRG1. PROTAC BRM/BRG1 degrader-1 can be used for cancer research. Blue: E3 ligase ligand (HY-168243), black: linker (HY-168244). Red: BRM/BRG1 inhibitor (HY-W539427)[1]. |
| CAS | 2724268-88-4 |
| Formula | C54H63N9O9S |
| Molar Mass | 1014.20 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Matthew Netherton, et al. Compounds and uses thereof. Patent. WO2021207291. |
PROTAC BRM/BRG1 degrader-1
CAS: 2724268-88-4 F: C54H63N9O9S W: 1014.20
PROTAC BRM/BRG1 degrader-1 (Example 253) is a PROTAC BRM/BRG1 degrader, with DC50 of 10-100 nM for BRM, > 1 μM for BRG1
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This product is for research use only, not for human use. We do not sell to patients.