| Bioactivity | PL-017 is a potent and selective μ opioid receptor agonist with an IC50 of 5.5 nM for 125I-FK 33,824 binding to μ site. PL-017 produces long-lasting, reversible analgesia in rats[1]. |
| Invitro | PL-017 has an IC50 of 10000 nM for 125I-DADLE binding to δ site[1]. |
| Name | PL-017 |
| CAS | 83397-56-2 |
| Shortening | YP-{N(Me)Phe}-P-NH2 |
| Formula | C29H37N5O5 |
| Molar Mass | 535.63 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |