| Bioactivity | PKMYT1-IN-2 is a potent PKMYT1 inhibitor with an IC50 of 5.7 nM. PKMYT1-IN-2 inhibits the growth of HCC1569 cells with an IC50 of 22 nM (WO2024061343A1; compound 2)[1]. |
| Target | IC50: 5.7 nM (PKMYT1) |
| CAS | 3033609-84-3 |
| Formula | C22H19N5O2 |
| Molar Mass | 385.42 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Dongxing Zhu, et al. Membrane-associated tyrosine and threonine kinase inhibitor and use thereof. WO2024061343A1. |