Bioactivity | PKMYT1-IN-1 (Compound 1) is an inhibitor for membrane-associated tyrosine and threonine kinase (PKMYT1), with an IC50 of 8.8 nM. PKMYT1-IN-1 inhibits proliferation of tumor cell HCC1569 with IC50 of 42 nM[1]. |
CAS | 3033609-83-2 |
Formula | C21H17N5O2 |
Molar Mass | 371.39 |
Transport | Room temperature in continental US; may vary elsewhere. |
Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
Reference | [1]. Zhu D, et al., Membrane-associated tyrosine and threonine kinase inhibitor and use thereof. WO2024061343A1. |