| Bioactivity | PKC-theta inhibitor is a selective PKC-θinhibitor, with an IC50 of 12 nM. | ||||||||||||
| Name | PKC-theta inhibitor | ||||||||||||
| CAS | 736048-65-0 | ||||||||||||
| Formula | C20H25F3N6O3 | ||||||||||||
| Molar Mass | 454.45 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
| Storage |
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| Reference | [1]. Cywin CL, et al. Discovery of potent and selective PKC-theta inhibitors. Bioorg Med Chem Lett. 2007 Jan 1;17(1):225-30. |