| Bioactivity | PKA-IN-1 is a potent and selective cyclic AMP-dependent protein kinase (PKA) catalytic subunit (cAK) inhibitor with an IC50 of 0.03 μM[1]. | |||||||||
| Target | IC50: 0.03 μM (cAK) | |||||||||
| Name | PKA-IN-1 | |||||||||
| CAS | 179985-52-5 | |||||||||
| Formula | C13H11N3O | |||||||||
| Molar Mass | 225.25 | |||||||||
| Appearance | Solid | |||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | |||||||||
| Storage |
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| Reference | [1]. Z X Lu, et al. Selective inhibition of cyclic AMP-dependent protein kinase by isoquinoline derivative. Biol Chem Hoppe Seyler. 1996 Jun;377(6):373-8 |