| Bioactivity | PF-4800567 hydrochloride is a potent and selective inhibitor of?casein kinase?1? (CK1?), with an?IC50?of 32 nM, which is greater than 20-fold selectivity over CK1δ (IC50, 711 nM). PF-4800567 hydrochloride is useful in probing unique roles between these two kinases in multiple signaling pathways[1]. |
| Target | IC50: 32 nM ((CK1?) |
| Name | PF-4800567 hydrochloride |
| CAS | 1391052-28-0 |
| Formula | C17H19Cl2N5O2 |
| Molar Mass | 396.27 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Walton KM, et al. Selective inhibition of casein kinase 1 epsilon minimally alters circadian clock period. J Pharmacol Exp Ther. 2009 Aug;330(2):430-9. |
PF-4800567 hydrochloride
CAS: 1391052-28-0 F: C17H19Cl2N5O2 W: 396.27
PF-4800567 hydrochloride is a potent and selective inhibitor of?casein kinase?1? (CK1?), with an?IC50?of 32 nM, which is
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