| Bioactivity | PE 22-28 is a TREK-1 inhibitor with IC50 value of 0.12 nM. PE 22-28 also is a 7 amino-acid peptide that is used as a core sequence for preparing analogs by chemical modifications and also by substitution of amino-acids. PE 22-28 can be used for the research of depression[1]. |
| Invitro | PE 22-28 displays good specificity and affinity for TREK-1 channel with IC50 value of 0.12 nM[1]. |
| Name | PE 22-28 |
| CAS | 1801959-12-5 |
| Shortening | GVSWGLR |
| Formula | C35H55N11O9 |
| Molar Mass | 773.88 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |