| Bioactivity | PDHK-IN-7 (compound 32) is an inhibitor of pyruvate dehydrogenase kinase with an IC50 value of 17 nM.PDHK-IN-7 activates PDH in rat livers and has a glucose-lowering effect in Zucker fatty rats[1]. |
| CAS | 1220965-73-0 |
| Formula | C20H17F3N2O2 |
| Molar Mass | 374.36 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Masafumi Inoue, et al. Design and synthesis of novel fluorene derivatives as inhibitors of pyruvate dehydrogenase kinase. Bioorg Med Chem Lett. 2024 Sep 1:109:129839. |
PDHK-IN-7
CAS: 1220965-73-0 F: C20H17F3N2O2 W: 374.36
PDHK-IN-7 (compound 32) is an inhibitor of pyruvate dehydrogenase kinase with an IC50 value of 17 nM.PDHK-IN-7 activates
Sales Email：peptidedb@qq.com
This product is for research use only, not for human use. We do not sell to patients.