| Bioactivity | PD 156252 is a hexapeptide that is a highly potent endothelin (ET) antagonist. PD 156252 has enhanced binding affinity for rabbit ETA and rat ETB receptor subtypes with IC50 values of 1.0 and 40 nM, respectively. |
| Name | PD 156252 |
| CAS | 175592-65-1 |
| Sequence | Ac-{d-Bhg}-Leu-Asp-Ile-{(N-Me)Ile}-Trp |
| Shortening | Ac-{d-Bhg}-LDI-{(N-Me)Ile}-W |
| Formula | C53H69N7O10 |
| Molar Mass | 964.16 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Cody WL, et al. Design of a potent combined pseudopeptide endothelin-A/endothelin-B receptor antagonist, Ac-DBhg16-Leu-Asp-Ile-[NMe]Ile-Trp21 (PD 156252): examination of its pharmacokinetic and spectral properties. J Med Chem. 1997 Jul 4;40(14):2228-40. |
PD 156252
CAS: 175592-65-1 F: C53H69N7O10 W: 964.16
PD 156252 is a hexapeptide that is a highly potent endothelin (ET) antagonist. PD 156252 has enhanced binding affinity f
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