Bioactivity | PCAF-IN-1 is a highly selective PCAF inhibitor. PCAF-IN-1 is a antitumor agents, which can be used in tumor treatment research[1]. | ||||||||||||
Invitro | PCAF-IN-1 (Compound 32) (10 μM, 72 hours; human tumor cell lines) exerts the most potent antitumor activities against human cancer cell lines[1]. Cell Cytotoxicity Assay[1] Cell Line: | ||||||||||||
Name | PCAF-IN-1 | ||||||||||||
CAS | 2439194-86-0 | ||||||||||||
Formula | C15H11ClN6 | ||||||||||||
Molar Mass | 310.74 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Turky A, et al. Design, synthesis, and antitumor activity of novel compounds based on 1,2,4-triazolophthalazine scaffold: Apoptosis-inductive and PCAF-inhibitory effects. Bioorg Chem. 2020 Aug;101:104019. |