| Bioactivity | PAR-2 antagonist 1 (Compound 9a) is a protease-activated receptor 2 (PAR2) antagonist with an IC50 value of 0.9 μM. PAR-2 antagonist 1 can effectively inhibit the proliferation and migration of breast cancer cells[1]. |
| Target | IC50: 0.9 μM (PAR2). |
| CAS | 313957-41-4 |
| Formula | C27H22N2O2 |
| Molar Mass | 406.48 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Kim T, et al. Discovery of Protease-activated receptor 2 antagonists derived from phenylalanine for the treatment of breast cancer. Bioorg Chem. 2024 Sep;150:107496. |
PAR-2 antagonist 1
CAS: 313957-41-4 F: C27H22N2O2 W: 406.48
PAR-2 antagonist 1 (Compound 9a) is a protease-activated receptor 2 (PAR2) antagonist with an IC50 value of 0.9 μM. PAR
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