| Bioactivity | P2X7 receptor antagonist-2 is a potent P2X7 receptor antagonist with a pIC50 value of 6.5-7.5. P2X7 receptor antagonist-2 has efficacy of combating neuroinflammation[1]. |
| Target | pIC50:6.5-7.5 (P2X7 receptor) |
| Name | P2X7 receptor antagonist-2 |
| CAS | 851269-75-5 |
| Formula | C19H18Cl2N2O2 |
| Molar Mass | 377.26 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Steadman JGA, et, al. 5-oxo-3-pyrrolidinecarboxamide derivatives as p2x7 modulators. WO2009077559A2 |