| Bioactivity | P2X4 antagonist-1 (Compound 24) is an antagonist for P2X4 with IC50 of 15 nM[1]. |
| CAS | 2055601-42-6 |
| Formula | C20H15Cl3N2O4S |
| Molar Mass | 485.77 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Reference | [1]. Werner S, et al., Discovery and characterization of the potent and selective P2X4 inhibitor N-[4-(3-Chlorophenoxy)-3-sulfamoylphenyl]-2-phenylacetamide (BAY-1797) and structure-guided amelioration of its CYP3A4 induction profile[J]. Journal of Medicinal Chemistry, 2019, 62(24): 11194-11217. |