Bioactivity | OGT-IN-2 (compound 4) is a potent O-GlcNAc transferase (OGT) inhibitor, with IC50 values of 30 and 53 μM for sOGT and ncOGT, respectively[1]. | ||||||||||||
Target | IC50: 30 ± 2 μM (sOGT), 53 ± 7 μM (ncOGT) | ||||||||||||
Name | OGT-IN-2 | ||||||||||||
CAS | 442665-87-4 | ||||||||||||
Formula | C23H27ClN2O3S | ||||||||||||
Molar Mass | 446.99 | ||||||||||||
Appearance | Solid | ||||||||||||
Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
Storage |
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Reference | [1]. Gross BJ, et al. Discovery of O-GlcNAc transferase inhibitors. J Am Chem Soc. 2005 Oct 26;127(42):14588-9. |