| Bioactivity | NaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7, exhibits 80-fold selectivity versus hNaV1.5[1]. | ||||||||||||
| Name | NaV1.7 inhibitor-1 | ||||||||||||
| CAS | 1494585-79-3 | ||||||||||||
| Formula | C23H30FNO4S | ||||||||||||
| Molar Mass | 435.55 | ||||||||||||
| Appearance | Solid | ||||||||||||
| Transport | Room temperature in continental US; may vary elsewhere. | ||||||||||||
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| Reference | [1]. Sun S, Identification of Selective Acyl Sulfonamide-Cycloalkylether Inhibitors of the Voltage-GatedSodium Channel (NaV) 1.7 with Potent Analgesic Activity. J Med Chem. 2019 Jan 24;62(2):908-927. |
NaV1.7 inhibitor-1
CAS: 1494585-79-3 F: C23H30FNO4S W: 435.55
NaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7
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